Small-molecule FRET probes for protein kinase activity monitoring in living cells.

In this study, the applicability of fluorescently labeled adenosine analogue-oligoarginine conjugates (ARC-Photo probes) for monitoring of protein kinase A (PKA) activity in living cells was demonstrated. ARC-Photo probes possessing subnanomolar affinity towards the catalytic subunit of PKA (PKAc) a...

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Autori principali: Vaasa, A, Lust, M, Terrin, A, Uri, A, Zaccolo, M
Natura: Journal article
Lingua:English
Pubblicazione: 2010