Mimics of L-rhamnose: Analogues of rhamnopyranose containing a constituent alpha-amino acid at the anomeric position. A rhamnopyranose analogue of hydantocidin

Mimics of L-rhamnose: Analogues of rhamnopyranose containing a constituent alpha-amino acid at the anomeric position. A rhamnopyranose analogue of hydantocidin

Ionic brominative oxidation of 2-amino derivatives of protected heptonolactones derived from L-rhamnose provides a key bicyclic intermediate for the synthesis of analogues of L-rhamnopyranose with spirohydantoins and spirodiketopiperazines at the anomeric position; the same intermediate can be used...

Полное описание

Библиографические подробности
Главные авторы:	Estevez, J, Smith, M, Wormald, MR, Besra, G, Brennan, P, Nash, R, Fleet, G
Формат:	Journal article
Опубликовано:	1996

Схожие документы

A galactopyranose analogue of hydantocidin
по: Brandstetter, T, и др.
Опубликовано: (1996)

Mimics of L-rhamnose: Anomeric spirohydantoins and diketopiperazines - Approaches to novel N-linked glycopeptides of rhamnofuranose
по: Estevez, J, и др.
Опубликовано: (1996)

Glucofuranose analogues of hydantocidin
по: Brandstetter, T, и др.
Опубликовано: (1996)

Divergent intermediates for the generation of libraries of L-rhamnose mimics
по: Smith, M, и др.
Опубликовано: (1996)

Mimics of L-rhamnose: Synthesis of C-glycosides of L-rhamnofuranose and an alpha-azidoester as divergent intermediates for combinatorial generation of rhamnofuranose libraries
по: Estevez, J, и др.
Опубликовано: (1996)

SPIRODIKETOPIPERAZINES AT THE ANOMERIC POSITION OF MANNOPYRANOSE - NOVEL N-LINKED GLYCOPEPTIDES INCORPORATING AN ALPHA-AMINO-ACID AT THE ANOMERIC POSITION OF MANNOPYRANOSE
по: Estevez, J, и др.
Опубликовано: (1995)

Spirodiketopiperazines of mannofuranose: carbopeptoid alpha-amino acid esters at the anomeric position of mannofuranose
по: Estevez, J, и др.
Опубликовано: (1998)

Inhibition of naringinase (L-rhamnosidase) by piperidine analogues of L-rhamnose: Scaffolds for libraries incorporating trihydroxypipecolic acids
по: Shilvock, J, и др.
Опубликовано: (1996)

A highly cytotoxic L-rhamnose analogue of the antitumour agent spicamycin
по: Martin, A, и др.
Опубликовано: (1998)

TRI-PEPTIDES AND TETRA-PEPTIDES INCORPORATING AN ALPHA-AMINO-ACID AT THE ANOMERIC POSITION OF MANNOFURANOSE
по: Estevez, J, и др.
Опубликовано: (1994)

TOWARDS 7 CARBON SUGAR MIMICS OF L-RHAMNOSE
по: Wheatley, J, и др.
Опубликовано: (1995)

Mirror image mimics of rhamnose fucose galactose and mannose
по: Shilvock, J, и др.
Опубликовано: (1997)

SPIROCYCLIC PEPTIDES AT THE ANOMERIC POSITION OF MANNOFURANOSE
по: Estevez, J, и др.
Опубликовано: (1994)

SPIROHYDANTOINS OF GLUCOFURANOSE - ANALOGS OF HYDANTOCIDIN
по: Brandstetter, T, и др.
Опубликовано: (1995)

KETALS OF L-RHAMNOHEPTONOLACTONES - POTENTIAL MIMICS OF L-RHAMNOSE
по: Wheatley, J, и др.
Опубликовано: (1994)

Synthesis and biological evaluation of enantiomeric rhamnose analogues of the antitumour agent spicamycin - is the mode of action by modification of N-linked glycoproteins?
по: Martin, A, и др.
Опубликовано: (1999)

ANOMERIC SPIROHYDANTOINS OF MANNOFURANOSE - APPROACHES TO NOVEL ANOMERIC AMINO-ACIDS BY AN OXIDATIVE RING CONTRACTION
по: Burton, J, и др.
Опубликовано: (1993)

Oxetane cis- and trans-beta-amino-acid scaffolds from L-rhamnose by efficient S(N)2 reactions in oxetane rings; pseudoenantiomeric analogues of the antibiotic oxetin
по: Johnson, S, и др.
Опубликовано: (2004)

Sugar amino acids at the anomeric position of carbohydrates: synthesis of spirocyclic amino acids of 6-deoxy-L-lyxofuranose
по: Bleriot, Y, и др.
Опубликовано: (2006)

Synthesis of bicyclic oxa- and aza-L-rhamnose mimics; Potential inhibitors of alpha-L-rhamnosidases
по: Pickering, L, и др.
Опубликовано: (1998)

POTENT INHIBITION OF GLYCOGEN-PHOSPHORYLASE BY A SPIROHYDANTOIN OF GLUCOPYRANOSE - FIRST PYRANOSE ANALOGS OF HYDANTOCIDIN
по: Bichard, C, и др.
Опубликовано: (1995)

Carbopeptoids: peptides and diketopiperazines incorporating the anomeric centre of mannopyranose
по: Long, D, и др.
Опубликовано: (2001)

6-deoxyhexoses from L-rhamnose in the search for inducers of the rhamnose operon: Synergy of chemistry and biotechnology
по: Liu, Z, и др.
Опубликовано: (2016)

Synthesis of Sulfo-Sialic Acid Analogues: Potent Neuraminidase Inhibitors in Regards to Anomeric Functionality
по: Christopher J. Vavricka, и др.
Опубликовано: (2017-08-01)

Inhibition of UDP-Gal mutase and mycobacterial galactan biosynthesis by pyrrolidine analogues of galactofuranose
по: Lee, R, и др.
Опубликовано: (1997)

Tetrahydrofuran alpha-azido esters: Precursors of anomeric alpha-amino acid monomers via radical bromination
по: Smith, M, и др.
Опубликовано: (1999)

(+)-MUSCARINE FROM L-RHAMNOSE
по: Mantell, S, и др.
Опубликовано: (1991)

MUSCARINE FROM L-RHAMNOSE
по: Mantell, S, и др.
Опубликовано: (1992)

Photobromination of a bicyclic mimic of alpha-L-fucose; Components for a combinatorial library of rigid fucose analogues
по: Smelt, K, и др.
Опубликовано: (1999)

A compendium of cyclic sugar amino acids and their carbocyclic and heterocyclic nitrogen analogues.
по: Risseeuw, M, и др.
Опубликовано: (2013)

3-HYDROXYMUSCARINES FROM L-RHAMNOSE
по: Mantell, S, и др.
Опубликовано: (1993)

Synthesis of the naringinase inhibitors L-swainsonine and related 6-C-methyl-L-swainsonine analogues: (6R)-C-methyl-L-swainsonine is a more potent inhibitor of L-rhamnosidase by an order of magnitude than L-swainsonine
по: Hakansson, A, и др.
Опубликовано: (2008)

Anomeric specificity of D-xylose isomerase.
по: Collyer, C, и др.
Опубликовано: (1992)

Sugar mimics from sugar lactones
по: Fleet, G, и др.
Опубликовано: (1998)

A PRACTICAL SYNTHESIS OF (+)-MUSCARINE FROM L-RHAMNOSE
по: Mantell, S, и др.
Опубликовано: (1992)

Synthesis of excitatory amino acid analogues
по: Goundry, W, и др.
Опубликовано: (2006)

An approach to the generation of simple analogues of the antitumour agent spicamycin.
по: Mons, S, и др.
Опубликовано: (2003)

The structural basis of the inhibition of human glycosidases by castanospermine analogues.
по: Winchester, BG, и др.
Опубликовано: (1990)

SPECIFIC-INHIBITION OF GLYCOGEN-PHOSPHORYLASE BY A SPIRODIKETOPIPERAZINE AT THE ANOMERIC POSITION OF GLUCOPYRANOSE
по: Krulle, T, и др.
Опубликовано: (1995)

Antimicrobial Activity of Amino Acid Analogues and Their Derivatives
по: Dácil Hernández, и др.
Опубликовано: (2017-10-01)