Synthesis of new 1,2-disubstituted benzimidazole analogs as potent inhibitors of Î-Glucuronidase and in silico study

Synthesis of new 1,2-disubstituted benzimidazole analogs as potent inhibitors of Î-Glucuronidase and in silico study

New benzimidazole analogues (1–18) were synthesized and characterized through different spectroscopic techniques such as 1H NMR, 13C NMR and HREI-MS. All analogues were screened for β-glucuronidase inhibitory potential. All analogues showed varied degree of inhibitory potentials with IC50 values ran...

Ամբողջական նկարագրություն

Մատենագիտական մանրամասներ
Հիմնական հեղինակներ:	Muhammad Taha, Ahmad Khan, Aftab, Rahim, Fazal, Imran, Syahrul, Mohammed Salahuddin, Uddin, Nizam, Mohammed Khan, Khalid, Ali Shah, Syed Adnan, Zafar, Ameeduzzafar, Zakaria, Zainul Amiruddin
Ձևաչափ:	Հոդված
Հրապարակվել է:	Elsevier B.V. 2021

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