Characterization of the Aquaporin-9 Inhibitor RG100204 In Vitro and in <i>db/db</i> Mice

Characterization of the Aquaporin-9 Inhibitor RG100204 In Vitro and in <i>db/db</i> Mice

Aquaporin-9 (AQP9) is a facilitator of glycerol and other small neutral solute transmembrane diffusion. Identification of specific inhibitors for aquaporin family proteins has been difficult, due to high sequence similarity between the 13 human isoforms, and due to the limited channel surface areas...

Πλήρης περιγραφή

Λεπτομέρειες βιβλιογραφικής εγγραφής
Κύριοι συγγραφείς:	Marilina Florio, Angelica Engfors, Patrizia Gena, Jessica Larsson, Alessandro Massaro, Stella Timpka, Martina Kvist Reimer, Per Kjellbom, Eric Beitz, Urban Johanson, Michael Rützler, Giuseppe Calamita
Μορφή:	Άρθρο
Γλώσσα:	English
Έκδοση:	MDPI AG 2022-10-01
Σειρά:	Cells
Θέματα:	membrane transport aquaglyceroporins metabolic homeostasis energy balance glycerol metabolism gluconeogenesis
Διαθέσιμο Online:	https://www.mdpi.com/2073-4409/11/19/3118

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